Home Tools
Log in
Cart

Search Result

Search Results for " vasopressin 1 "

20

Compounds

Cat No. Product Name Synonyms Targets
T21296 Desmopressin acetate trihydrate Desmogalen,Adiuretin,Deamino Arginine Vasopressin,Vasopressin 1-Desamino-8-arginine
Desmopressin acetate is a synthetic replacement for vasopressin, which reduces urine production. Medical use of Desmopressin acetate includes: (a) bed wetting; (b) diabetes insipidus; (c) nighttime urination; (d) clottin...
T2568 Felypressin Octapressin,Felypressin Acetate,PLV-2,H-[Cys-Phe-Phe-Gln-Asn-Cys]-Pro-Lys-Gly-NH2 Vasopressin Receptor
Felypressin (Octapressin) is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activity.
T64174 Vasopressin V2 receptor antagonist 1
Vasopressin V2 receptor antagonist 1 (Compound 4g) is a vasopressin V2receptor (V2R) antagonist (Ki: 3.8 nM). dominant polycystic kidney disease (ADPKD).
T2568L Felypressin acetate 2-(L-Phenylalanine)-8-L-lysinevasopressin,PLV2. H-Cys-Phe-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2 (Disulfide bond),PLV 2,PLV-2 Vasopressin Receptor
Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures.
T7284 Argipressin acetate (113-79-1(free base)) Others
Vasopressin acetate is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth muscle...
T14494 Balovaptan RG7314 Vasopressin Receptor
Balovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors. It is used for the research of autism.
T6288 Mozavaptan OPC31260l,OPC-31260 Vasopressin Receptor
Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
T80197 Vasopressin Dimer (parallel) (TFA) Vasopressin Receptor
Vasopressin Dimer (parallel) TFA, a parallel dimer of Vasopressin, has the capability to activate four G protein-coupled receptors—namely, V1aR, V1bR, V2R, and OTR [1].
T76510 [Asu1,6-Arg8]Vasopressin
[Asu1,6-Arg8]Vasopressin is a vasopressin agonist that enhances cyclic AMP accumulation and adrenocorticotropic hormone (ACTH) release triggered by corticotropin-releasing factor (CRF) in cultured rat anterior pituitary ...
T83488 [Lys8] Vasopressin Desglycinamide
[Lys8] Vasopressin Desglycinamide, a vasopressin analog, supports the maintenance of active and passive avoidance behavior and aids in the facilitation of memory consolidation processes [1].
T76633 (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin
(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin, a potent vasopressin V1 receptor (VP V1R) antagonist, significantly lowers mean arterial pressure (MAP) in rats [1].
T76573 [8-L-arginine] deaminovasopressin
[8-L-arginine] deaminovasopressin (dAVP) is a vasopressin analog [1] .
T80073 Dp[Tyr(methyl)2,Arg8]-Vasopressin Vasopressin Receptor
Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].
T83502 [Deamino-4-valine, 8-D-arginine]-Vasopressin dVDAVP
[Deamino-4-valine, 8-D-arginine]-Vasopressin (dVDAVP) is a highly potent and specific antidiuretic agent, exhibiting prolonged effects [1] [2].
T80198 Vasopressin Dimer (anti-parallel) (TFA) Vasopressin Receptor
Vasopressin Dimer (anti-parallel) TFA, an anti-parallel dimer form of vasopressin, has the capability to activate four G protein-coupled receptors: V1aR, V1bR, V2R, and OTR [1].
T76509 Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potent agonist at the pituitary corticotrope receptor [1].
T75834 Antagonist G TFA
Antagonist G TFA is a potent antagonist of vasopressin, with additional, weaker antagonistic effects on GRP and Bradykinin. This compound also promotes AP-1 transcription and enhances cellular sensitivity to chemotherapy...
T79173 PF-06478939 Oxytocin Receptor
PF-06478939 is a peptide that functions as an agonist at the oxytocin (OT) receptor and vasopressin receptor without crossing the blood-brain barrier. It exhibits EC50 values of 0.01 nM at the OT receptor and 0.078 nM at...
T80270 Invopressin OCE-205 Vasopressin Receptor
Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in research related to cirrhosis conditions such as bacterial peritonitis, HRS2, and refractory ascites [1].
T80137 (d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin d(CH2)5[Tyr(Me)2, Dab5]AVP Vasopressin Receptor
(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].

Compounds

Desmopressin acetate trihydrate
T21296
Synonym: Desmogalen,Adiuretin,Deamino Arginine Vasopressin,Vasopressin 1-Desamino-8-arginine
Target:
Felypressin
T2568
Synonym: Octapressin,Felypressin Acetate,PLV-2,H-[Cys-Phe-Phe-Gln-Asn-Cys]-Pro-Lys-Gly-NH2
Target: Vasopressin Receptor
Vasopressin V2 receptor antagonist 1
T64174
Synonym:
Target:
Felypressin acetate
T2568L
Synonym: 2-(L-Phenylalanine)-8-L-lysinevasopressin,PLV2. H-Cys-Phe-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2 (Disulfide bond),PLV 2,PLV-2
Target: Vasopressin Receptor
Argipressin acetate (113-79-1(free base))
T7284
Synonym:
Target: Others
Balovaptan
T14494
Synonym: RG7314
Target: Vasopressin Receptor
Mozavaptan
T6288
Synonym: OPC31260l,OPC-31260
Target: Vasopressin Receptor
Vasopressin Dimer (parallel) (TFA)
T80197
Synonym:
Target: Vasopressin Receptor
[Asu1,6-Arg8]Vasopressin
T76510
Synonym:
Target:
[Lys8] Vasopressin Desglycinamide
T83488
Synonym:
Target:
(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin
T76633
Synonym:
Target:
[8-L-arginine] deaminovasopressin
T76573
Synonym:
Target:
Dp[Tyr(methyl)2,Arg8]-Vasopressin
T80073
Synonym:
Target: Vasopressin Receptor
[Deamino-4-valine, 8-D-arginine]-Vasopressin
T83502
Synonym: dVDAVP
Target:
Vasopressin Dimer (anti-parallel) (TFA)
T80198
Synonym:
Target: Vasopressin Receptor
Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
T76509
Synonym:
Target:
Antagonist G TFA
T75834
Synonym:
Target:
PF-06478939
T79173
Synonym:
Target: Oxytocin Receptor
Invopressin
T80270
Synonym: OCE-205
Target: Vasopressin Receptor
(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
T80137
Synonym: d(CH2)5[Tyr(Me)2, Dab5]AVP
Target: Vasopressin Receptor
1 2
TargetMol